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Biological EvaluationFacile SynthesisEnantioselective SynthesisFunctional GroupRegioselective SynthesisDipolar CycloadditionMichael AdditionDIASTEREOSELECTIVE SYNTHESISClick ChemistryAsymmetric SynthesisGreen ChemistryRoom TemperatureIntramolecular CouplingNatural ProductsCoupling ReactionsMulticomponent ReactionsSynthetic OrganicDrug DiscoveryMetal-free SynthesisHeterocyclic Compounds